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.., .. .: , 2008. 224 c.
ISBN 978-5-9704-0578-9
( ): pharmazeutischewirkstoffe1982.djvu
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DBP 1168 910 (Beecham; Anm. 3,7.1962; GB-Prior. 21.7.1961).
USP 3 144445 (AmericanHome; ert. 11.8.1964; Anm. 26.12.1962).
DAS 1445 506 (Bristol-Myers; Anm. 24.10.1963; USA-Prior. 29.10.1962).
DAS 1 545 534 (Astra; Anm. 4.3.1965; S-Prior. 6.3.1964).
DAS 2029 195 (Yamanouchi; Anm. 13.6.1970; J-Prior. 16.6.1969).
DAS 1 800 698 (American Home Products; Anm. 2.10.1968; USA-Prior. 2.10.1967). DOS 2 755 903 (Dobfar;Anm. 15.12.1977; I-Prior. 16.12.1976).
Enzymatische und mikrobiologische Verfahren:
USP 3 079307 (Bayer; ert. 26.2.1963; D-Prior. 7.10.1961).
DBP 1966 521 (Kyowa Hakko; Anm. 9.9.1969; J-Prior. 18.9.1968, 8.10.1968).
DAS 1 967 074 (Kyowa Hakko; Anm. 9.9.1969; J-Prior. 18.9.1968, 8.10.1968).
DAS 2 050 983 (Kyowa Hakko; Anm. 16.10.1970; J-Prior. 16.10.1969).
USP 4073 687 (Shionogi; ert. 14.2.1978; J-Prior. 14.5.1975).
Ampicillin-Salze:
DBP 1 197 460 (Bayer; Anm. 4.9.1962).
DOS 1670 111 (Bristol-Myers; Anm. 16.7.1966).
DBP 1 670191 (Beecham; Anm. 24.2.1967; GB-Prior. 3.3.1966).
DAS 1795 129 (Beecham; Anm. 14.8.1968; USA-Prior. 18.8.1967).
DBP 1 903 388 (American Home Products; Anm. 23.1.1969; USA Prior. 23.1.1968). DAS 2 623 835 (Boehringer Ing.; Anm. 28.5.1976).
Trihydrat:
USP 3 157 640 (Bristol-Myers; ert. 17.11.1964; Anm. 21.3.1963).
Ampicillio
52 A Ampicillin - Anagestonacetat
D: Amblosin® (Hoechst)
Ampicillin (ratiopharm) Ampi-Tablinen® (Sanorania) Binotal® (Bayer)
Cymbi® (Dolorgiet)
Deripen® (Schering) Dura-Ampicillin (Durachemte) Lucipen® (Hoechst)-Komb. Pen-Bristol® (Griinenthal) Penbrock® (Beecham)
Suractin® (Lappe)
F: Ampicil® (Arkodex)
Penbritine® (Beecham-Sevigne) Penicline (Delagrange)
Prototapen (Bristol)
Totapen® (Bristol)
Ukapen® (Spret-Mauchant)
GB: Amfipen® (Brocades)
Penbritin® (Beecham)
I: Ampen® (Medosan)
Ampibeta® (Violam-Farma vigor) Ampibiotic® (Ottolenghi)
Ampicil® (Ausonia)
Ampicillina Pharmax® (Pharmax) Ampicillina Pierrel® (Pierrel) Ampicina® (Sigmatau)
Ampifen® (Intersint)
Ampilan® (Ibirn)
Ampilisa® (Lisaphanna)
Ampilux® (Tubi Lux Farma) Ampisint® (Proter)
Ampitex® (Neopharmed) Ampivax® (Ripari-Gero) Amplenil® (Orma) Amplibios®(Panther-Osfa Chemie) Amplicid® (Cifa)
Amplipen® (Labif)
Amplipenyl® (Isf)
Ampliscocil® (Ici)
Amplital® (Farmitalia)
Ampiizer® (Off)
Anidropen® (Wyeth)
Anticyl® (San Cario)
Axgocillina® (Beta)
Binotal® (Bayer)
Bio-Ampi® (Donatello)
Biocellina® (Magis)
Citicil® (Ct)
Eurocillin® (Borromeo) Farmampil® (Gazzini)
Geycillina® (Geymonat) Gramcil/ma® (Caber)
LampociJlina® Orale (Sidus)
Napicil® (Montefarmaco)
Overcillina® (Archifar)
Fen-Ampil® (Nuovo Cons. Sanit. Naz.) Penberm® (Bergamon Soc. It.)
Penisint B.G.® (Boniscontro & G.) Pentrexil® (Bristol Ital. Sud)
Platocillina® (Crosara)
Principen® (Squibb)
Radiocillina® (Radiumfarma)
Saicil® (Libra)
Sernabiotic® (Libra)
Sesquiciliina® (Ita)
Sintopenyl® (Aesculapius)
Totalciclina® (Benvegna) zahlreiche Komb.-Praparate J: Acucillin®(Fuji)-Komb.
Adobaciliin® (Tobisbi)
Amipenix® (Toyo Jozo)
Ampicillin (Nihon Iyakuhin; Pfizer-Taito; Sanko; Sawai; Showa Shinyaku;
Tatsumi; Toho; Towa; Tsuruhara) Bionacillin® (Takata)
Bonapicillin® (Taiho)
Cilleral® (Bristre-Banyu)
Combipenix® (Toyo Jozo)-Komb. Domicillin® (Marupi)
Isodllin® (Kanto)
Ohtecin® (Kyowa)
Penbritin® (Beecham-Fujisawa)
Penimic® (SS Seiyaku)
Pentrex® (Banyu)
Pharcillin® (Toyo Pharmar)
Solcillin® (Takeda)-Komb.
Synpenin® (Sankyo)
Tokiocillin® (Isei)
Totacillin® (Beecham)
Totaclox® (Beecham)-Komb.
Viccillin® (Meiji)
USA: Alpen® (Lederle)
Amcill® (Parke Davis)
Omnipen® (Wyeth)
Pen-А® (Pfizer)
Penbritin® (Ayerst)
Pensyn® (Upjohn)
Polycillin® (Squibb)
Principen® (Squibb)
О 1 Damp® (Mallincrodt) SK-Ampicillin™ (Smith Kline 4- French) Totacillin® (Beecham-Massengill)
Anagestonacetat 3137-73-3 Gestagen
2740-52-5 Anageston
17-hydroxy-6a-methyJpregn-4-en-20-one-ace.tate
Anagestonacetat - Ancitabin A 53
+ hs-ch2-ch2-sh
3 20-Dioxo-17-hydroxy- 1,2-Ethandithiol
6^-methyl-i-pregnen
[Fyridir • HC1 j Pyriditiium-
chiorid
1. Ra-Ni/C2HsOH 2 CHjCOOH/(CH*COIiO !
1. Rarwy-Nickel
2. Essigsaure/Essigsaureanhydnd/ p-fcluolsulfcnsaur*
Belg-P 624370 (Ortho; Anm. 31.10.1962; USA-Prior. 6-6.1962, 24.7.1961; F-Prior. 23.7.1962). USA: Anatropin® (Ortho)
Ancitabin
(Cycloxytidine)
31698-14-3
10212-25-6 Hydrochlorid
Antileucamicum;
Cytostaticum
(2R,1',RS'nS^)-iR)-233a,9a-tetrahydro-3-hvdroxv 6-immn 6/7 !uro-[2',3' ;4.5 o4azaki[Г>,^-(j)
pyrimidine-2-methanol
NHz
O^N'
HOCH, +
я
P0C13
НгО/СН}СООС2Н5
HO OH Cytidm
Phosphor-
oxychlorid
DOT 12,304(1976).
T. Kanai et al., Chem. Pharm. Bull. 18,2569 (1970). Weitere Verfahren:
E. R. Walwick et al., Proc. Chem. Soc. (London) 1959, 84. L. L. Doerr, J. J. Fox, J. Org. Chem. 31,1465 (1967).
W. V. Ruyle, T. Y. Shenn, J. Med. Chem. 10,331 (1967). К. K. Kugawa, M. Ichino, Tetrahedron Lett. 1970, 867.
J:
Cyclo-C (Kohjin)
54 A Androstanolon - Anetholtrithion
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