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* pregna-l,4-diene-3,20-dione,l l,21-dihydroxy-l7-[(l-oxopentyl)oxy]-,(l l/3)-21-acetate
HO-CH4 HO-CH2v n
1. Рќ,РЎ-(РЎРќРіР-РЎ(РЎРЎРќСЌ)Р· / H3C-<^_>-S03H
2. HCI/CH3OH
1 Orthovaleriansauretnmethylester
0-РЎ0-(РЎРќ2)Р·-РЎРќР·
Prednisolon-17-valerat
Prednivalacetat - Prednyliden P 757
(CH3CO)20/Pyr>din
Prednivalacetat
DOT 15,421 (1979).
R. Gardi et al., Gazz. Chim. Ital. 93,431 (1963).
Prednisolon-17-valerat:
DBP 1214677 (Francesco Vismara; Anm. 1.6.1962; I-Prior. 24.6.1961). USP 3 147 249 (Francesco Vismara; ert. 1.9.1964; I-Prior. 13.6.1961). vgl. auch Hydrocortisonbutyrat, Betametasonvalerat.
I: AceprevalВ® (Parke-Davis-Vister)
Prednyliden 599-33-7 Glucocorticoid
11Р”17,21 -trihydroxy-16-methylenepregna-1,4-diene-3,20-dione
Р—/Р-Acstoxy- 16-methyl- 20-oxo-5,16-pregnadien
758 P Prednyliden - Prednyliden-diethyl-aminoacetat - Pregnenolon
DBP 1 134 074 (E. Merck AG; Anm. 31.1.1959).
H. J. Mannhardt et al., Tetrahedron Lett. 1960, 21.
D. Taub et al., J. Org. Chem. 25, 2258 (1960).
Weiteres Verfahren:
USP 3 068 226 (Merck & Co.; ert. 1962; Prior. 1961,1959).
D: DecortilenВ® (Merck) I: DacortiEenВ® Merck (Bracco)
F: DecortileneВ® (Farmex)
Prednyliden-diethyl- 6890-42'2 Glucocorticoid aminoacetat 22887-42-9 Hydrochlorid
llftl7,21-trihydroxy-16-methylenpregna-l,4-diene-3,20-dione-21-diethylaminoacetate но—ch,
[(H5C2l2N-CH2-C0]20
Oiethylaminoessigsaure-
anhydrid
[ Pyridin
(HsC2)2N - CH2- CO-O-CH2.
Prednyliden-diethylaminoacetat
DBP 1 134 074 (E. Merck AG; Anm. 31.1.1959). Kombination mit Chinolin-Derivaten:
Belg-P 829 197 (Grosjean; Anm. 16.5.1975).
D: DecortilenВ® sol. (Merck)
Pregnenolon 145-13-1 Glucocorticoid
4598-67-8 Succinat 1778-02-5 Acetat
3-hydroxypregn-5-ene-20-one
Pregnenolon - Prenyiamin - Pridinol P 759
H3C-C0-0 )6 - Dehydropregnenoicn- 3/5- acetat
1 H2/Pd
2 Hydrolyse
Ehr hart- Ruschig, III, 341.
Ullmann, 3. Auflage, Bd. 8, 664, und dort zitierte Literatur. Weitere Verfahren:
Ullmann, 3. Auflage, Bd. 8, 660.
The Merck Index, 7533 (Rahway 1976) und dort zitierte Literatur.
F: FadiamoneВ® Creme (Sauba)-Komb.-Acetat USA: Formula 405 (Doak)-Succinat
PanzaloneВ® (Doak)-Succinat PrenolonВ® (Schering)
Prenyiamin
390-64-7 69-43-2 Lactat 21156-48-9 Gluponat
Coronarvasodilatator
<V-(3,3-diphenylpropyl)-a-methylphenethylamine
Q
РЎ
6
РќР·РЎ\ h2/f
ch-ch2-ch2-nh2 + /СЂ~РЎРќ2~\_}
Рѕ
3,3-Oiphenylpropylamin
Phenylaceton
'Q
Prenyiamin
DBP 1 111 642 (Hoechst; Anm. 7.5.1958). DBP 1 100 031 (Hoechst; Anm. 7.5.1958).
D: DaxautenВ® (Woelm Pharma)
SegontinВ® (Hoechst)
SegontinВ®-Digoxin (Hoechst)-Komb.
F: ClemodrilВ® (Hoechst)-Komb.
SegontineВ® (Hoechst)
GB: SynadrinВ® (Hoechst)
I: AngiovigorВ® (Violani-Farmavigor) AngorsanВ® (Isola-Ibi)
Corditin-SameВ® (Savoma)
EucardionВ® (Vita)
IncoranВ® (Ita)
IrrorinВ® (Alfa Farm.)
ReocorinВ® (Farmochimica Itai.) SegontinВ® (Hoechst) WasangorВ® (Wassermann) CrepasinВ® (Hoei)
EpocolВ® (Teisan-Nagase) HerzconВ® (Sana)
LactamineВ® (Daisan)
NP 30 (Sanken)
OnleminВ® (Ono)
PrectofactВ® (Showa Yakuhin) Prenylamine Lactate (Towa) RoininВ® (Mohan)
SegontinВ® (Hoechst)
Pridinol
511-45-5
968-58-1
6856-31-1
Hydrochlorid
Methansulfonat
Anticholinergicum;
Antiparkinson-Mittel
a,a-diphenyl-l-piperidinepropanol
760 P Pridinol - Prilocain - Primaperon
<Qh-MgBr ♦ )-сн2-сн2-0
h5c2o
Phenylmagn#- 3-Piper id inopropjonsaure-smmbronVid bzw ethyiester Srombenzol
OH
РЁ -CH2-CH2-
6
<0
^~^-CO~CH3 + (CH20)„ + Hl/^>
Acetophenon
Paraform- Piperidin aidehyd
0_^CH2_CH2-,q
w-pipendinopropiophenon
Om
Bromberaol bzw Phenylmagnssium-
DBP875 660 (Hoechst; Anm. 1941).
D: Lyseen-HommelВ® (Hommel) ParKSВ® 12 (Hommel F: PARKS-12В® (Laroze)
I: AlgolisinaВ® (Bonomelli-Hommel) LyseenВ® (Bonomelli-Hommel)
HikicenonВ® (Tatsumi) KonlaxВ® (Nippon Shinyaku) LoxeenВ® (Maniko-Tobishi) MitanolineВ® (Toyo Pharmar) TrilaxВ® (Toyo Seiyaku Kasei)
Prilocain
721-50-6
1786-81-8
Hydrochloric!
Lokalanastheticum
2-' propvlannno) Рѕ propionotolnidiile
CH3
0-NH
CH3
I
o-Toluidin
2-8rompropionyl-
bromid
CH3
^ NH—CO—CH—Br
CH3
h2n-c3h7
DOT 3,65(1967).
GB-P 839943 (Astra; Anm. 6-6.1958; S-Prior. 26.6.1957).
N. Lofgren, C. Tegner; Acta Chem. Scand. 14,486,490 (1960).
/=( РЎРќР· | <r^-NH-CO-CH-NH-C3H7 1
Prilocain
D: XylonestВ® (Astra)
F: CitanestВ® Rachianesthesie (Roger Beilon) GB; CitanestВ® (Astra)
I: CitanestВ® (Dentalica)-Komb. J: CitanesrВ® (Astra-Fujisawa) USA. CitanestВ® (Astra)
Primaperon 15847-48-0
4'-fluoro-4-piperidinobutyrophenone
Vasodilatator
Primaperon - Primidon - Probenecid P 761
F-<Q^C-CH2-CH2-CH2-Cl * HN^> -* ; f-^-C-CHz-CHj-CHz-N^
0 I 0
I
w-Chlor-4-fluorbutyrophenon Piperidin j_Primaperon
FP 1 301 863 (Science Union; Anm. 29.6.1961).
FP 1 459M (ScienceUnion; Anm. 18.8.1961; Prior. 29.6.1961).
F: DiviatorВ® (Servier)-Komb.
Primidon 125-33-7 Antiepilepticum
(Primadone)
5-ethyldihydro-5-phenyl-4,6( I H,5 /-/)pynmicinedione nh2
o^c
H=c-c.c.NH2
65
Ethylphenyl-
malonsaurediamid
